Chapter 1 Uptake Transporters of the Human OATP Family

Chapter 2 In Vitro and In Vivo Evidence of the Importance of Organic Anion Transporters (OATs) in Drug Therapy

Chapter 3 Organic Cation Transporters (OCTs, MATEs), In Vitro and In Vivo Evidence for the Importance in Drug Therapy

Chapter 4 Drug Transporters

Chapter 5 The Role of the Sodium-Taurocholate Cotransporting Polypeptide (NTCP) and of the Bile Salt Export Pump (BSEP) in Physiology and Pathophysiology of Bile Formation

Chapter 6 P-glycoprotein: Tissue Distribution, Substrates, and Functional Consequences of Genetic Variations

Chapter 7 Importance of P-glycoprotein for Drug–Drug Interactions

Chapter 8 Multidrug resistance proteins (MRPs, ABCCs): importance for pathophysiology and drug therapy.

Chapter 10 Molecular Mechanisms of Drug Transporter Regulation

Chapter 11 In Vivo Probes of Drug Transport: Commonly Used Probe Drugs to Assess Function of Intestinal P-glycoprotein (ABCB1) in Humans